產(chǎn)品編號(hào) | D51433 |
英文名稱 | Hydroxyfasudil HCl |
中文名稱 | |
別 名 | ROCK抑制劑 |
克 隆 號(hào) | |
CAS | 155558-32-0 |
理論分子量 | 343.83 kDa |
檢測(cè)分子量 | |
性 狀 | Lyophilized |
保存條件 | Store in dry, dark place for one year. |
注意事項(xiàng) | This product as supplied is intended for research use only, not for use in human, therapeutic or diagnostic applications. |
產(chǎn)品介紹 |
Hydroxyfasudil, aslo known as HA1100, is a cell-permeable hydroxylated metabolite of HA-1077, is a potent inhibitor of Rho-associated kinase (ROCK) (Ki = 150 nM). Hydroxyfasudil alleviates demyelination through the inhibition of MOG antibody and microglia activation in cuprizone mouse model. |