| 產(chǎn)品編號(hào) | D51420 |
| 英文名稱 | GSK180736A |
| 中文名稱 | |
| 別 名 | ROCK1/GRK2抑制劑 |
| 克 隆 號(hào) | |
| CAS | 817194-38-0 |
| 理論分子量 | 365.36 kDa |
| 檢測(cè)分子量 | |
| 性 狀 | Lyophilized |
| 保存條件 | Store in dry, dark place for one year. |
| 注意事項(xiàng) | This product as supplied is intended for research use only, not for use in human, therapeutic or diagnostic applications. |
| 產(chǎn)品介紹 |
GSK180736A is potent and selective inhibitor of GRK2 with an IC50 of 0.77 μM25 and >100-fold selectivity over other GRKs. It is a weak inhibitor of PKA with an IC50 of 30 μM, but highly potent against ROCK1 (IC50 = 100 nM). |
