| 產(chǎn)品編號(hào) | D51373 |
| 英文名稱 | K-252a |
| 中文名稱 | |
| 別 名 | PKA/PKC/CaMKII抑制劑 |
| 克 隆 號(hào) | |
| CAS | 99533-80-9 |
| 理論分子量 | 467.47 kDa |
| 檢測(cè)分子量 | |
| 性 狀 | Lyophilized |
| 保存條件 | Store in dry, dark place for one year. |
| 注意事項(xiàng) | This product as supplied is intended for research use only, not for use in human, therapeutic or diagnostic applications. |
| 產(chǎn)品介紹 |
K-252a, also known as SF 2370, is an alkaloid isolated from Nocardiopisis bacteria. This staurosporine analog is a highly potent cell permeable inhibitor of CaM kinase and phosphorylase kinase (IC50 = 1.8 and 1.7 nmol/L, respectively). At higher concentrations it is also an efficient inhibitor of serine/threonine protein kinases (IC50 of 10 to 30 nmol/L). |
